PT141 (BREMELANOTIDE) 10MG

Description

⚠ For laboratory research use only. Not for human consumption.

CAS NO: 1607799-13-2

Molecular Formula: C₅₀H₆₈N₁₄O₁₀

Molecular Weight: 1,025.16 g/mol

Form: Lyophilized powder

Appearance: white powder

Storage: 2-8°

Purity: ≥99%

PT-141 (Bremelanotide) is a synthetic peptide that acts on the melanocortin receptor system in the brain. Unlike medications such as Viagra or Cialis that primarily affect blood flow, PT-141 works through the central nervous system and is studied for its effects on sexual desire and arousal. involved in sexual motivation and arousal rather than directly increasing blood flow. as the brand-name product , was approved by the FDA in 2019 for treating acquired, generalized HSDD in premenopausal women.

PT-141 MECHANISM OF ACTION: ADVANCED NEUROLOGICAL PATHWAYS

PT-141 exerts its effects through sophisticated melanocortin receptor interactions:

• Selective Receptor Activation: Demonstrates high affinity for MC4R (Melanocortin 4 Receptor)with significant activity at MC3R, while showing minimal activity at MC1R, MC2R, and MC5R (Hadley, 2005)
• Blood-Brain Barrier Penetration: Crosses the blood-brain barrier efficiently due to its small molecular size and lipophilic properties, enabling direct central nervous system effects (King et al., 2007)
• Dopaminergic Pathway Modulation: Indirectly influences dopamine release in the nucleus accumbensthrough melanocortin receptor activation, affecting motivation and reward pathways (Martin et al., 2011)
• Nitric Oxide Activation: Stimulates nitric oxide synthase activityin specific neural circuits, contributing to its physiological effects (Rosen et al., 2013)

EXPERIMENTAL PREPARATION

For accurate research application:

1. Reconstitutewith appropriate volume of bacteriostatic water
2. Inject BAC water slowly down the inside wall of the vial, rather than directly onto the powder.
3. Gently swirluntil fully dissolved (do not vortex)
4. Administerimmediately or store at 4°C protected from light
5. Reconstituted: Stable 30 days at 4°C

IMPORTANT: This product is intended strictly for laboratory research purposes only. NOT for human or animal consumption. NOT for medical or diagnostic use. These products have not undergone evaluation by the U.S. Food and Drug Administration. By purchasing, you confirm compliance with all applicable regulations.